释义 |
Anordrin 基本例句 双炔失碳酯,53号抗孕片 Anordrinhas first been synthesized and developed in China in 1970’s .双炔失碳酯,是70年代我国自行研制的甾体避孕药物,开始曾试用于抗早孕,随后将它改作探亲避孕药。 Objective: To find anordrin analogs possessing higher bioactivity and lower side effect after reconstructing anordrin.目的:通过改造双炔失碳酯的化学结构,获得活性更高、副作用更小的避孕药。The relative binding affinities of four steroid hormonal drugs for estrogen receptors of uterine cytosol were detemined by competitive binding assay and shown to be in the following order: ethinyl ostradiol>estradiol>anordrin>danazol. 根据;E_2和E_R具有高度专一性及亲和力的特性,应用竞争性试验比较了炔雌醇、雌二醇、双炔失碳酯、丹那唑与兔子宫胞液雌激素受体的相对结合亲和力;KeywordsAnordrin;Analogue;Antifertility activity;双炔失碳酯;类似物;抗生育活性; KeywordsAnordrin;Chorion;Decidua;Endocrine function;双炔失碳酯;绒毛;蜕膜;内分泌功能; |